Synthesis of the esters of 1-alkyl-2-aminoindolyl-3-acetic acids by the Kost reaction

Authors

  • В. П. Жестков All-Russian Scientific Center for the Safety of Biologically Active Substances (VNTs BAV), Kupavna, Moscow Oblast, 142450
  • В. Г. Забродная All-Russian Scientific Center for the Safety of Biologically Active Substances (VNTs BAV), Kupavna, Moscow Oblast, 142450
  • А. И. Чернышев All-Russian Scientific Center for the Safety of Biologically Active Substances (VNTs BAV), Kupavna, Moscow Oblast, 142450

Abstract

The reaction of the esters of N-alkyl-N-phenylhydrazinocarbonylpropionic acids with phosphorus oxychloride in dioxane or with phosgene in benzene leads to the formation of the esters of 1-alkyl-2-aminoindolyl-3-acetic acids and of the corresponding N-alkyl-N-phenylaminosuccinimides.

How to Cite
Zhestkov, V. P.; Zabrodnaya, V. G.; Chernyshev, A. I. Chem. Heterocycl. Compd. 1995, 31, 1302. [Khim. Geterotsikl. Soedin. 1995, 1502.]

For this article in the English edition, see DOI https://doi.org/10.1007/BF01168624

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Published

1995-11-25

Issue

No. 11 (1995)

Section

Original Papers