SUBSTITUTED AND SPIRO-ANNELATED PERHYDRO-1,2,3-OXATHIAZINE 2,2-DIOXIDES AND 1-BENZYL-4-METHYLAZETIDINES

Authors

  • A. V. Varlamov Russian People's Friendship University, Moscow 117198
  • N. V. Sidorenko Russian People's Friendship University, Moscow 117198
  • F. I. Zubkov Russian People's Friendship University, Moscow 117198
  • A. I. Chernyshev Russian People's Friendship University, Moscow 117198
  • K. F. Turchin Center for Drug Chemistry/All-Russian Scientific Research Pharmaceutical Chemistry Institute, Moscow 119815

Keywords:

azetidines, homoallyl amines, 1,2,3-oxathiazine 2,2-dioxides

Abstract

We obtained perhydro-1,2,3-oxathiazine 2,2-dioxides by cyclization of 4-N-benzylamino-4-tetramethylene(phenyl-, methylphenyl-, dimethyl)but-1-enes in conc. H2SO4 at 25°C. When treated with an alcoholic solution of base, the oxathiazines are converted to 2-substituted and spiro-annelated 1-benzyl-4-methylazetidines.

How to Cite
Varlamov, A. V.; Sidorenko, N. V.; Zubkov, F. I.; Chernyshev, A. I.; Turchin, K. F. Chem. Heterocycl. Compd. 2004, 40, 1097. [Khim. Geterotsikl. Soedin. 2004, 1261.]

For this article in the English edition, see DOI 10.1023/B:COHC.0000046704.43034.bd

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Published

2004-08-25

Issue

No. 8 (2004)

Section

Original Papers