CONVERSION OF 2-AMINOMETHYLBENZOTHIAZOLES INTO IMIDAZO[5,1-<i>b</i>]BENZOTHIAZOLES

Authors

  • В. B. Авидон Ordzhonikidze All-Union Chemical-Pharmaceutical Scientific Research Institute, Moscow
  • M. Н. Щукина Ordzhonikidze All-Union Chemical-Pharmaceutical Scientific Research Institute, Moscow

DOI:

https://doi.org/10.1007/141

Abstract

A number of substituted 2-aminomethylbenzothiazoles are synthesized. The corresponding ureas or thioureas are also obtained by reaction with arylisocyanates or arylisothiocyanates. Heating the substituted ureas or thioureas at temperatures above their melting points cyclizes them to 9-substituted 2-hydroxy- or 2-mercaptoimidazo[5,1-b]benzothiazoles, which are derivatives of a new heterocyclic system.

Authors: V. V. Avidon, M. N. Shchukina.

English Translation in Chemistry of Heterocyclic Compounds, 1965, 1 (1), pp 42-45

http://link.springer.com/article/10.1007/BF01168917

Published

2013-01-09

Issue

No. 1 (1965)

Section

Original Papers