HETEROCYCLIZATIONS OF α-HETEROATOM-SUBSTITUTED ORGANOBORONATES

Authors

  • Oleksandr O. Grygorenko Enamine Ltd., 78 Chervonotkatska St., Kyiv 02094 Taras Shevchenko National University of Kyiv, 60 Volodymyrska St., Kyiv 01601
  • Yevhen M. Ivon Enamine Ltd., 78 Chervonotkatska St., Kyiv 02094 Taras Shevchenko National University of Kyiv, 60 Volodymyrska St., Kyiv 01601

DOI:

https://doi.org/10.1007/5517

Keywords:

organoboron compounds, heterocyclization, nitrogen-containing heterocycles, azoles, metathesis

Abstract

Heterocyclizations of boronates bearing a heteroatom-containing substituent at theα-position are reviewed. Synthesis of heteroaromatic boronates by heterocyclizations of nitrogen- and oxygen-containing compounds (e.g., aldehydes, ketones, or epoxides) bearing a boronate moiety, as well as preparation of (partially) saturated heterocyclic derivatives via metathesis reactions are discussed.

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Published

2020-02-28

Issue

Vol. 56 No. 2 (2020)

Section

Heterocycles in Focus