SYNTHESIS OF PYRIMIDO[1,2-<i>a</i>]INDOLES

Authors

  • Игорь Л. Никонов Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, 22/20 Sofiiy Kovalevskoi St., Yekaterinburg 620219, Russia
  • Дмитрий С. Копчук Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, 22/20 Sofiiy Kovalevskoi St., Yekaterinburg 620219, Russia
  • Григорий В. Зырянов Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, 22/20 Sofiiy Kovalevskoi St., Yekaterinburg 620219, Russia
  • Владимир Л. Русинов Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St., Yekaterinburg 620002, Russia Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, 22/20 Sofiiy Kovalevskoi St., Yekaterinburg 620219, Russia

DOI:

https://doi.org/10.1007/6341

Abstract

This review considers methods for the synthesis of pyrimido[1,2-a]indoles and their ring-fused derivatives, covering publications from the last 10 years. Depending on the synthons used for assembling the target structure, three main approaches to the synthesis of pyrimido[1,2-a]indoles can be distinguished: annulation of a pyrimidine ring to 2-aminoindoles, modification of other indole derivatives, and miscellaneous methods.

 

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Published

2021-10-21

Issue

Vol. 57 No. 10 (2021)

Section

Heterocycles in Focus