TETRAHYDROAZEPINES WITH AN ANNULATED FIVE-MEMBERED HETEROAROMATIC RING

Authors

  • Иванна Ю. Данилюк Institute of Organic Chemistry, National Academy of Sciences of Ukraine, 5 Akademika Kukhara St., Kyiv 02094
  • Мыхайло В. Вовк Institute of Organic Chemistry, National Academy of Sciences of Ukraine, 5 Akademika Kukhara St., Kyiv 02094

DOI:

https://doi.org/10.1007/6847

Keywords:

furoazepines, imidazoazepines, isothiazoloazepines, isoxazoloazepines, oxazoloazepines, pyrazoloazepines, pyrroloazepines, thiazoloazepines, thienoazepines, triazoloazepines

Abstract

The review summarizes and analyzes the literature data on the synthetic design of promising biologically active hydrogenated furo-, thieno-, pyrrolo-, and azoloazepine systems. The information is systematized according to the principle of prevalence and significance of the employed synthetic methods: annulation of an azepine ring to a five-membered heteroaromatic ring, annulation of a five-membered heteroaromatic ring to an azepine ring, ring expansion reactions of hetaro-annulated cyclohexanones and piperidines. The bibliography of the review contains 94 sources published in 2000–2022.

Authors: Ivanna Yu. Danyliuk*, Mykhailo V. Vovk

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Published

2022-11-16

Issue

Vol. 58 No. 11 (2022)

Section

Review Articles